PKM2-IN-9
PKM2-IN-9 (compound C1) is a potent inhibitor of PKM2, with the inhibition rate of 75% at 50 μM. PKM2-IN-9 plays an important role in cancer research[1].
Product Specifications
CAS Number
[498568-75-5]
UNSPSC
12352005
Target
Pyruvate Kinase
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Cancer
Smiles
O=C(C1=CC=CC=C1)NCC2=NC3=C(N2CC(NC4=CC=CC(C)=C4)=O)C=CC=C3
Molecular Formula
C24H22N4O2
Molecular Weight
398.46
References & Citations
[1]Beth Israel Deaconess Medical Center. Pyruvate kinase M2 inhibitors and methods using them for the treatment of disease. World Intellectual Property Organization, WO2008019139 A2 2008-02-14
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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