Telapristone acetate
Telapristone acetate (CDB-4124) is a potent progesterone receptor (PR) modulator. Telapristone acetate inhibits the proliferation of ovarian cancer cells by inducing cell cycle arrest and apoptosis. Telapristone effectively inhibits the occurrence and development of spontaneous and chemically induced mammary tumors in rats. Telapristone acetate can be used for breast and ovarian cancer research[1][2].
Product Specifications
CAS Number
[198414-31-2]
Product Name Alternative
CDB-4124
UNSPSC
12352005
Target
Apoptosis; CDK; PARP; Progesterone Receptor
Related Pathways
Apoptosis; Cell Cycle/DNA Damage; Epigenetics; Vitamin D Related/Nuclear Receptor
Field of Research
Cancer; Endocrinology
Solubility
10 mM in DMSO
Smiles
C[C@@]12[C@](CC[C@]2(OC(C)=O)C(COC)=O)([H])[C@@]3([H])C([C@@H](C4=CC=C(N(C)C)C=C4)C1)=C(CC5)C(CC3)=CC5=O
Molecular Formula
C31H39NO5
Molecular Weight
505.65
References & Citations
Shipping Conditions
Room temperature
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-16483/
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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