Gintemetostat
Gintemetostat (KTX-1001) is a potent NSD2 inhibitor with an IC50 ranging from 0.001 μM to 0.01 μM. As a piperidinyl-methyl-purineamine derivative, gintemetostat has potential applications in cancer research[1].
Product Specifications
CAS Number
[2604513-16-6]
Product Name Alternative
KTX-1001
UNSPSC
12352005
Target
Histone Methyltransferase
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Purity
99.81
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
FC(C=C(C(F)=C1)OC)=C1C2=NC=C(N3C[C@](N)(CCC3)[C@H](O)C(F)F)C(CN4C5=NC=NC(N)=C5N=C4)=C2
Molecular Formula
C25H26F4N8O2
Molecular Weight
546.52
References & Citations
[1]Roberts M F, et al. 6-Methoxyflavonols from Brickellia veronicaefolia (compositae) [J]. Phytochemistry, 1980, 19 (1) : 127-129.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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