VUF5207

VUF5207, an Impentamine (HY-107564) analogue, is a partial agonist of histamine H3 receptor[1].

Product Specifications

CAS Number

[397248-39-4]

UNSPSC

12352005

Target

Histamine Receptor

Related Pathways

GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

Field of Research

Inflammation/Immunology

Smiles

N1=CNC(=C1)CCCCCN(C)C

Molecular Formula

C10H19N3

Molecular Weight

181.28

References & Citations

[1]Schihada H, et al. Development of a Conformational Histamine H3 Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists. ACS Sens. 2020 Jun 26;5 (6) :1734-1742.|[2]Soudijn W, et al. Structure-activity relationships of inverse agonists for G-protein-coupled receptors. Med Res Rev. 2005 Jul;25 (4) :398-426.