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HIF-1α-IN-6

Product Specifications

Target

HIF/HIF Prolyl-Hydroxylase

Related Pathways

Chromatin/Epigenetic|||Metabolism

Bioactivity

HIF-1?-IN-6 (compound 3s) is a potent inhibitor of HIF-1? with IC50 values of 0.6 nM and 53.3 nM in MiaPaCa-2 and MDA-MB-231 cells, respectively, and it suppresses HIF-1? expression by reducing HIF-1? mRNA levels [1].

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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