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CI-988 hemihydrate

Product Specifications

Target

Cholecystokinin Receptor

Related Pathways

GPCR/G Protein

Bioactivity

CI-988 hemihydrate (PD134308) is a potent and selective orally active CCK2R (cholecystokinin 2 receptor) antagonist, with an IC50 of 1.7 nM for mouse cortical CCK2. It is over 1600 times more selective for CCK2 than for CCK1 receptors. CI-988 hemihydrate exhibits anxiolytic and antitumor properties.

Molecular Formula

C35H42N4O6.1/2H2O

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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