RJG-2051
Product Specifications
CAS Number
2851993-77-4
Target
Reductase
Related Pathways
Metabolism|||Endocrinology/Hormones
Bioactivity
RJG-2051 is a selective covalent inhibitor of aldo-keto reductase family 1 member C3 (AKR1C3), with an IC50 value of 13 nM. It interferes with the metabolism of substrates such as androgens, estrogens, and prostaglandins through AKR1C3. RJG-2051 holds potential for cancer research.
Smiles
O=C(C1=CC=C(C=C1)S(=O)(=O)N2N=C(N=C2)C3CCCCC3)N4CCN(C=5C=CC=CC5OC)CC4
Molecular Formula
C26H31N5O4S
Molecular Weight
509.62
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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