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BGC4

Product Specifications

Target

Apoptosis

Related Pathways

Apoptosis

Bioactivity

BGC4 is a gold (III) complex based on biphenyl. It inhibits human recombinant thioredoxin reductase (TrxR) with an IC50 of 10.7 ?M, exhibits cytotoxicity with an IC50 of 5.4 ?M in MDA-MB-231 cells, and induces apoptosis. Additionally, BGC4 demonstrates antitumor activity in mouse models.

Molecular Formula

C30H32AuClF3N3

Molecular Weight

724.01

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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