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K 0859

BGG463 can inhibit c-ABL-T334I, BCR-ABL and BCR-ABL-T315I variants with a 50% inhibitory concentration (IC50) of 0.25 μM, 0.09 μM and 0.590 μM, respectively.

Product Specifications

CAS Number

890129-26-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

578.6

Molecular Formula

C30H29F3N6O3

Notes

Research use only, not for human use.

Receptor

C-ABL-T334I|Abl|Abl (T315I)

Available Sizes

Curated Selection

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