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Cilengitide

Cilengitide is a potent integrin inhibitor for αvβ3 receptor and αvβ5 receptor with IC50 of 4.1 nM and 79 nM in cell-free assays, respectively; ~10-fold selectivity against gpIIbIIIa. Phase 2.

Product Specifications

CAS Number

188968-51-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

588.66

Molecular Formula

C27H40N8O7

Notes

Research use only, not for human use.

Receptor

ΑVβ3 integrin| αVβ5 integrin

Available Sizes

Curated Selection

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