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ARS-853

ARS-853 is a mutant-specific, covalent inhibitor of KRAS (G12C) ; engages KRASG12C in biochemical assay with a rate constant of 76 M-1s-1.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

432.9437

Molecular Formula

C22H29ClN4O3

Notes

Research use only, not for human use.

Receptor

Ras

CAS Number

1629268-00-3

Available Sizes

Curated Selection

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