MS012
MS012 is a selective GLP inhibitor (IC50=7 nM) . MS012 can be used in research of GLP dysregulation, including cancer, inflammatory diseases, and neuroregenerative disorders[1].
Product Specifications
CAS Number
[2089617-83-2]
UNSPSC
12352005
Target
GLP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Cancer; Inflammation/Immunology; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ms012.html
Purity
98.9
Solubility
10 mM in DMSO
Smiles
COC1=CC2=NC(NCCCCCC)=NC(NC3CCN(CC3)C)=C2C=C1OC
Molecular Formula
C22H35N5O2
Molecular Weight
401.55
References & Citations
[1]Xiong Y, et al. Discovery of Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase. J Med Chem. 2017 Mar 9;60 (5) :1876-1891.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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