Vasopressin V2 receptor antagonist 2
Product Specifications
UNSPSC Description
Vasopressin V2 receptor antagonist 2 (Compound 33) is an antagonist of the arginine vasopressin V2 receptor (V2R) with a Ki value of 6.2 nM. Vasopressin V2 receptor antagonist 2 can effectively reduce cAMP levels, thereby inhibiting the growth of renal cysts[1].
Target Antigen
Vasopressin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/vasopressin-v2-receptor-antagonist-2.html
Solubility
10 mM in DMSO
Smiles
NC([C@@H](NC([C@@H](NC([C@@H]1CCCN1C([C@H](CC)NC([C@@H](NC([C@@H](NC([C@H](CC2=CC=C(C=C2)F)NC([C@@H](CC3=CC=C(OCC)C=C3)NC(CC4=CC=C(C=C4)C(C)(C)C)=O)=O)=O)C(C)C)=O)CC(N)=O)=O)=O)=O)CCCNC(N)=N)=O)CCCNC(N)=N)=O
Molecular Weight
1255.48
References & Citations
[1]Xiong X, et al. Long-Residence Time Peptide Antagonist for the Vasopressin V<sub>2</sub> Receptor to Treat Autosomal Dominant Polycystic Kidney Disease. J Med Chem. 2024;67(7):5935-5944.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-162394/Vasopressin-V2-receptor-antagonist-2-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-162394/
Clinical Information
No Development Reported
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