5-HT4 antagonist 1
5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6.
Product Specifications
CAS Number
[261766-73-8]
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/5-HT4_antagonist_1.html
Purity
98.95
Solubility
DMSO : 20 mg/mL (ultrasonic; warming; adjust pH to 3 with HCl; heat to 60°C)
Smiles
O=C(C1=C2OCCOC2=CC=C1)NCC3CCN(CCCS(=O)(N4CCN(C)CC4)=O)CC3
Molecular Formula
C23H36N4O5S
Molecular Weight
480.62
References & Citations
[1]Clark RD, et al. Identification of a 5-HT4 receptor antagonist clinical candidate through side-chain modification. Bioorg Med Chem Lett. 2005 Mar 15;15 (6) :1697-700.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
Apolipoprotein D
Available Sizes
Curated Selection
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