CDK9-IN-10

CDK9-IN-10 is a potent CDK9 inhibitor. CDK9-IN-10 is the ligand for the PROTAC CDK9 degrader-2 (HY-112811)[1].

CDK; Ligands for Target Protein for PROTAC

Reference compound

Cell Cycle/DNA Damage;PROTAC

Cancer

https://www.medchemexpress.com/cdk9-in-10.html

98.00

DMSO : ≥ 100 mg/mL

OC1=C2C(C(C=C(C3=CC=CC=C3)O2)=O)=C(O)C=C1OCC4=CC=CC=C4

360.36

[1]Bian J, et al. Discovery of Wogonin-based PROTACs against CDK9 and capable of achieving antitumor activity. Bioorg Chem. 2018 Dec;81:373-381.

Room Temperature

4°C (Powder, sealed storage, away from moisture and light)

http://file.medchemexpress.com/batch_PDF/HY-130850/CDK9-IN-10-DataSheet-MedChemExpress.pdf

http://file.medchemexpress.com/batch_PDF/HY-130850/CDK9-IN-10-SDS-MedChemExpress.pdf

No Development Reported

3542-63-0