BIM-23056 (TFA)
Product Specifications
UNSPSC Description
BIM 23056 TFA, a linear octapeptide, is a potent sst3 and sst5 somatostatin receptor antagonist with Ki values of 10.8, 5.7, respectively[1].
Target Antigen
Somatostatin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein;Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/bim-23056-tfa.html
Solubility
H2O
Smiles
OC(C(F)(F)F)=O.OC(C=C1)=CC=C1C[C@H](NC([C@@H](NC([C@H](N)CC2=CC=CC=C2)=O)CC3=CC=CC=C3)=O)C(N[C@@H](C(N[C@@H](CCCCN)C(N[C@@H](C(C)C)C(N[C@H](C(N[C@@H](C(N)=O)CC4=CC5=C(C=CC=C5)C=C4)=O)CC6=CC=CC=C6)=O)=O)=O)CC7=CNC8=CC=CC=C78)=O
Molecular Weight
1346.49
References & Citations
[1]Y C Patel, et al. Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5). Endocrinology. 1994 Dec;135(6):2814-7.|[2]W Feniuk, et al. Further evidence from functional studies for somatostatin receptor heterogeneity in guinea-pig isolated ileum, vas deferens and right atrium. Br J Pharmacol. 1995 Jul;115(6):975-80.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-P1203A/BIM-23056-TFA-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-P1203A/
Clinical Information
No Development Reported
CAS Number
1426173-61-6
Curated Selection
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