YEATS4-IN-1
YEATS4-IN-1 (Compound 4d) is a potent and selective YEATS4 binder that binds to the KAc recognition site of the YEATS structural domain with a Ki value of 33 nM[1].
Product Specifications
CAS Number
[3034365-92-6]
Product Name Alternative
PFI-8
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/yeats4-in-1.html
Solubility
10 mM in DMSO
Smiles
OC1(CN2C[C@H](C)[C@@H](C3=C(C=CC(C(NCC)=O)=C4)N4N=C3C)CC2)CCCCC1
Molecular Formula
C24H36N4O2
Molecular Weight
412.57
References & Citations
[1]Allyn T Londregan, et al. Discovery of High-Affinity Small-Molecule Binders of the Epigenetic Reader YEATS4. J Med Chem. 2023 Jan 12;66 (1) :460-472.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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