L-817818

L-817818 is a potent and subtype-selective agonist of the somatostatin receptor. L-817818 provides a direct approach to defining somatostatin receptor physiological functions[1]

Product Specifications

CAS Number

[217480-27-8]

UNSPSC

12352005

Target

Somatostatin Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Endocrinology

Assay Protocol

https://www.medchemexpress.com/l-817818.html

Purity

99.80

Solubility

DMSO : 54 mg/mL (ultrasonic; warming)

Smiles

C[C@H](N)COC([C@@H](CCCCN)NC(CC1=C(C2=CC3=C(C=CC=C3)C=C2)NC4=C1C=CC5=CC=CC=C45)=O)=O

Molecular Formula

C33H36N4O3

Molecular Weight

536.66

References & Citations

[1]Rohrer SP, et al. Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry [published correction appears in Science 1998 Nov 27;282 (5394) :1646]. Science. 1998;282 (5389) :737-740.