α-helical CRF 9-41 acetate

Product Specifications

Target

CRFR

Related Pathways

GPCR/G Protein

Purity

0.966

Bioactivity

?-helical CRF 9-41 acetate is a competitive antagonist of CRF2 (KB = 100 nM) and a partial agonist of CRF1 (EC50 = 140 nM) .

Smiles

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