RVD-Hp?

N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM) .

C([C@@H](NC([C@@H](NC([C@H](CCCNC(=N)N)N)=O)C(C)C)=O)CC(O)=O)(=O)N1[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC2=CC=CC=C2)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC3=CN=CN3)C(O)=O)=O)CO)=O)CC(C)C)=O)CC(C)C)=O)CCCCN)=O)=O)CC(N)=O)=O)C(C)C)=O)CCC1