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Rucaparib camsylate

Product Specifications

CAS Number

1327258-57-0

Target

PARP|||Others

Related Pathways

DNA Damage/DNA Repair|||Others|||Chromatin/Epigenetic

Bioactivity

Rucaparib (AG014699) camsylate is an orally active inhibitor of PARP proteins (PARP-1, PARP-2, and PARP-3) with a Ki=1.4 nM for PARP-1, and also inhibits hexose hexaphosphate dehydrogenase (H6PD) . Rucaparib camsylate has potential for investigation in debulking resistant prostate cancer (CRPC) studies.

Molecular Formula

C19H18FN3O.xC10H16O4S

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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