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Axl-IN-9

Product Specifications

CAS Number

2487649-73-8

Target

Others|||TAM Receptor

Related Pathways

Tyrosine Kinase/Adaptors|||Others

Bioactivity

Axl-IN-9 is a potent inhibitor of AXL (IC50: 26 nM) with excellent transmembrane properties.Axl-IN-9 exhibits good pharmacokinetic properties in animals.Axl-IN-9 can be used to study proliferative, autoimmune, allergic, transplant rejection, inflammatory, cancer or other mammalian diseases.

Smiles

NC1=C2C(=CN(C)C2=NC=N1)C3=CC=C(NC(=O)C=4C(=O)N(N(C)C4C)C5=CC=CC=C5)C=C3

Molecular Formula

C25H23N7O2

Molecular Weight

453.5

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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