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CDK4/6-IN-9

Product Specifications

CAS Number

2688098-02-2

Target

CDK|||Others

Related Pathways

Cell Cycle/Checkpoint|||Others

Bioactivity

CDK4/6-IN-9 (compound 10) is a selective inhibitor of CDK4/6, demonstrating activity on CDK6/cyclin D1 (IC50: 905 nM), and holds potential research value in multiple myeloma (MM) .

Smiles

FC=1C(C=2C=3C(N(C)C2)=NC=CC3)=NC(NC4=CC=C(CN5CCNCC5)C=N4)=NC1

Molecular Formula

C22H23FN8

Molecular Weight

418.47

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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