TRPV1 antagonist 3
Product Specifications
Target
Others|||TRP/TRPV Channel
Related Pathways
Membrane transporter/Ion channel|||Others
Bioactivity
TRPV1 antagonist 3 (Compound 7q) is a highly potent TRPV1 receptor antagonist with an IC50 of 2.66 nM against capsaicin. It exhibits selectivity in its mode of action, is orally bioavailable (60%), and can penetrate the central nervous system [1].
Molecular Formula
C23H25N3OS
Molecular Weight
391.53
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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