BRD4 Inhibitor-15
Product Specifications
CAS Number
2761366-60-1
Target
Bcl-2 Family|||Epigenetic Reader Domain|||c-Myc|||Caspase|||Apoptosis|||Others
Related Pathways
Others|||Proteases/Proteasome|||Chromatin/Epigenetic|||Apoptosis|||Cell Cycle/Checkpoint
Bioactivity
BRD4 Inhibitor-15 (compound 13) is a highly potent and specific BRD4 inhibitor with an IC50 of 18 nM, inducing apoptosis in 22RV1 cells by regulating Bcl-2/Bax proteins and activating caspase-3 signaling, and down-regulating c-Myc levels, making it valuable for prostate cancer research [1].
Smiles
C(N1C=2C(=CC=C(C2)C=3C(OCC)=CC(=O)N(C)C3)C=N1)C4=CC=CC=C4
Molecular Formula
C22H21N3O2
Molecular Weight
359.42
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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