P-gp inhibitor 1
Product Specifications
CAS Number
2050747-49-2
Target
P-gp
Related Pathways
Neuroscience|||Membrane transporter/Ion channel
Purity
0.9865
Bioactivity
P-gp inhibitor 1 inhibits reversing P-glycoprotein-mediated multidrug resistance with an EC50 of 57.9 nM (K562/A02 cells) .
Smiles
COc1cc2CCN(CCc3ccc(Nc4nc(nc5ccccc45)-c4ccncc4)cc3)Cc2cc1OC
Molecular Formula
C32H31N5O2
Molecular Weight
517.62
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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