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GFB-8438

Product Specifications

CAS Number

2304549-73-1

Target

TRP/TRPV Channel

Related Pathways

Membrane transporter/Ion channel

Purity

0.9958

Bioactivity

GFB-8438 is a potent and subtype selective inhibitor of TRPC5 (IC50s of 0.18 and 0.29 ?M of hTRPC5 and hTRPC4, respectively) .

Smiles

FC(F)(F)c1ccccc1CN1CCN(CC1=O)c1cn[nH]c(=O)c1Cl

Molecular Formula

C16H14ClF3N4O2

Molecular Weight

386.76

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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